Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04148
Ion Channel
Glutamate receptor ionotropic subunit NMDA 1
Peptide Function
Antagonist
Gene Name
Grin1
Activity Data (nM)
IC50
93 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
NH2-GEQQVAKMAAQLARQNIAKGCKVNCYPCOOH
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
Con-R
Peptide Species
Conus radiatus (Rayed cone)
Peptide Name
Not available
CAS Number
Not available
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
Not specified
Temperature
25 °C
Test Method
Binding assay ([3H]MK-801 )
Test Species
Not specified
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
i-GluRs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available